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CAS RN: 85118-33-8 | 产品编码: G0405
Gaboxadol Hydrochloride
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| 产品编码 | G0405 |
| 纯度/分析方法 | >98.0%(HPLC) |
| 分子式/分子量 | C__6H__8N__2O__2·HCl = 176.60 |
| 外观与形状（20°C） | 固体 |
| 储存温度 | 室温 (15°C以下阴凉干燥处) |
| 包装和容器 | 25MG-Glass Bottle with Plastic Insert （查看图片） |
| CAS RN | 85118-33-8 |
| 相关CAS RN | 64603-91-4 |
| Reaxys-RN | 6534899 |
| PubChem物质ID | 253659629 |
| Merck Index (14) | 4321 |
| MDL编号 | MFCD00055180 |
技术规格
| Appearance | White to Almost white powder to crystal |
| Purity(HPLC) | min. 98.0 area% |
| Elemental analysis(Nitrogen) | 15.40 to 16.30 % |
物性（参考值）
| 熔点 | 236 °C |
GHS
相关法规
| RTECS# | NY3398000 |
运输信息
| HS编码* | 2934.99-000 |
应用
Gaboxadol Hydrochloride: A γ-Aminobutyric Acid Subtype A (GABAA) Receptor Agonist
Gaboxadol hydrochloride, also known as THIP, is a direct-acting γ-aminobutyric acid subtype A (GABAA) receptor agonist. GABAA receptor is widely considered to be an important target for most clinically effective sedative-hypnotic compounds. However, the clinical development program for gaboxadol was discontinued in 2007. (The product is for research purpose only.)
References
- Pharmacological characterization of a novel cell line expressing human α4β3δ GABAA receptors
- GABAA receptor α4 subunits mediate extrasynaptic inhibition in thalamus and dentate gyrus and the action of gaboxadol
- An extrasynaptic GABAA receptor mediates tonic inhibition in thalamic VB neurons
- Gaboxadol - a new awakening in sleep(a review)
- GABAA agonists and partial agonists: THIP (Gaboxadol) as a non-opioid analgesic and a novel type of hypnotic(a review)
- Development and validation of a selective and sensitive bioanalytical procedure for the quantitative determination of gaboxadol in human plasma employing mixed mode solid phase extraction and hydrophilic interaction liquid chromatography with tandem mass spectroscopic detection
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