Maximum quantity allowed is 999
Please select the quantity
CAS RN: 168273-06-1 | Product Number: R0205
Rimonabant
×
Purity: >98.0%(HPLC)
Synonyms:
- 5-(4-Chlorophenyl)-1-(2,4-dichlorophenyl)-4-methyl-N-(piperidin-1-yl)-1H-pyrazole-3-carboxamide
- SR 141716
Product Documents:
| Size | Unit Price | Saitama (Kawaguchi) | Hyogo (Amagasaki) | Stock in other WH |
Shipping Information
|
|---|---|---|---|---|---|
| 25MG |
¥25,100
|
It can be shipped in about 2-3 business days after ordering | It can be shipped from Saitama warehouse in about 2-3 business days after ordering | ≥40 | |
| 100MG |
¥75,200
|
It can be shipped in about 2-3 business days after ordering | It can be shipped from Saitama warehouse in about 2-3 business days after ordering | 14 |
* Available Stock: Prompt shipment (for products) in Saitama/Hyogo warehouse. Stock In Other WH: Shipment in about 2-3 Business Days from Saitama warehouse. Please contact us
if you need further information.
* The displayed price is the unit price and does not include consumption tax. The unit prices displayed are the latest and are subject to change without notice.
* To send your quote request for bulk quantities, please click on the "Request Bulk Quote" button. Please note that we cannot offer bulk quantities for some products.
*TCI frequently reviews storage conditions to optimize them. Please note that the latest information on the storage temperature for the products is described on our website.
* The displayed price is the unit price and does not include consumption tax. The unit prices displayed are the latest and are subject to change without notice.
* To send your quote request for bulk quantities, please click on the "Request Bulk Quote" button. Please note that we cannot offer bulk quantities for some products.
*TCI frequently reviews storage conditions to optimize them. Please note that the latest information on the storage temperature for the products is described on our website.
| Product Number | R0205 |
Purity / Analysis Method 
|
>98.0%(HPLC) |
| Molecular Formula / Molecular Weight | C__2__2H__2__1Cl__3N__4O = 463.79 |
| Physical State (20 deg.C) | Solid |
| Storage Temperature
|
Frozen (-20°C) |
| Store Under Inert Gas | Store under inert gas |
| Condition to Avoid | Air Sensitive,Heat Sensitive |
| CAS RN | 168273-06-1 |
| Reaxys Registry Number | 7231571 |
| PubChem Substance ID | 468592783 |
| MDL Number | MFCD04034714 |
Specifications
| Appearance | White to Almost white powder to crystal |
| Purity(HPLC) | min. 98.0 area% |
| NMR | confirm to structure |
Properties (reference)
GHS
| Pictogram |
|
| Signal Word | Warning |
| Hazard Statements | H361 : Suspected of damaging fertility or the unborn child. H371 : May cause damage to organs. H373 : May cause damage to organs through prolonged or repeated exposure. |
| Precautionary Statements | P501 : Dispose of contents/ container to an approved waste disposal plant. P260 : Do not breathe dust. P270 : Do not eat, drink or smoke when using this product. P202 : Do not handle until all safety precautions have been read and understood. P201 : Obtain special instructions before use. P264 : Wash skin thoroughly after handling. P280 : Wear protective gloves/ protective clothing/ eye protection/ face protection. P308 + P311 : IF exposed or concerned: Call a POISON CENTER/doctor. P405 : Store locked up. |
Related Laws:
| RTECS# | UQ6279632 |
Transport Information:
Application
Rimonabant: A Dual Inhibitor of Acyl CoA (cholesterol acyltransferase: ACAT) -1 and 2
Rimonabant and its hydrochloride [R0293] are also dual inhibitors of acyl-CoA (ACAT) 1 and 2, which catalyzes the intracellular synthesis of cholesteryl esters. (The product is for research use only.)
Reference
- Rimonabant is a dual inhibitor of acyl CoA:cholesterol acyltransferases 1 and 2
- Selective inhibition of sucrose and ethanol intake by SR 141716, an antagonist of central cannabinoid (CB1) receptors
- Keynote review: Medicinal chemistry strategies to CB1 cannabinoid receptor antagonists
- The psychiatric side-effects of rimonabant
- Development and validation of a high-performance liquid chromatographic method for bioanalytical application with rimonabant
Application
Rimonabant: A Selective Cannabinoid-1 Receptor (CB1) Antagonist.
Rimonabant (SR141716) is a selective cannabinoid-1 receptor (CB1) antagonist. CB1 is a G protein-coupled cannabinoid receptor that are found in the nervous system, and the body uses it to control food intake. It has been reported that rimonabant can help mammals to reduce food intake and to lose weight by blocking CB1 receptors. In clinical, rimonabant was withdrawn in 2008 due to serious psychiatric side effects. (The product is for research purpose only.)
References
Product Documents (Note: Some products will not have analytical charts available.)
Safety Data Sheet (SDS)
Please select Language.
The requested SDS is not available.
Please Contact Us for more information.
Specifications
C of A & Other Certificates
Please enter Lot Number
Incorrect Lot Number. Please input only the 4-5 alphanumeric characters before the hyphen.
Sample C of A
This is a sample C of A and may not represent a recently manufactured lot of the product.
A sample C of A for this product is not available at this time.
Analytical Charts
Please enter Lot Number
Incorrect Lot Number. Please input only the 4-5 alphanumeric characters before the hyphen.
The requested analytical chart is not available. Sorry for the inconvenience.