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CAS RN: 183232-66-8 | Product Number: A3151
AM 251
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Purity: >97.0%(HPLC)
Synonyms:
- 1-(2,4-Dichlorophenyl)-5-(4-iodophenyl)-4-methyl-N-(piperidin-1-yl)-1H-pyrazole-3-carboxamide
Product Documents:
| Size | Unit Price | Saitama (Kawaguchi) | Hyogo (Amagasaki) | Stock in other WH |
Shipping Information
|
|---|---|---|---|---|---|
| 50MG |
¥54,500
|
27 | 1 | Contact Us |
* Available Stock: Prompt shipment (for products) in Saitama/Hyogo warehouse. Stock In Other WH: Shipment in about 2-3 Business Days from Saitama warehouse. Please contact us
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* The displayed price is the unit price and does not include consumption tax. The unit prices displayed are the latest and are subject to change without notice.
* To send your quote request for bulk quantities, please click on the "Request Bulk Quote" button. Please note that we cannot offer bulk quantities for some products.
*TCI frequently reviews storage conditions to optimize them. Please note that the latest information on the storage temperature for the products is described on our website.
| Product Number | A3151 |
| Purity / Analysis Method | >97.0%(HPLC) |
| Molecular Formula / Molecular Weight | C__2__2H__2__1Cl__2IN__4O = 555.24 |
| Physical State (20 deg.C) | Solid |
| Storage Temperature | Frozen (<0°C) |
| Condition to Avoid | Heat Sensitive |
| CAS RN | 183232-66-8 |
| Reaxys Registry Number | 7780333 |
| PubChem Substance ID | 354335179 |
| MDL Number | MFCD01861181 |
Specifications
| Appearance | White to Light yellow powder to crystal |
| Purity(HPLC) | min. 97.0 area% |
| Elemental analysis(Nitrogen) | 9.60 to 10.60 % |
| NMR | confirm to structure |
Properties (reference)
| Melting Point | 196 °C |
GHS
| Pictogram |
|
| Signal Word | Warning |
| Hazard Statements | H315 : Causes skin irritation. H319 : Causes serious eye irritation. |
| Precautionary Statements | P264 : Wash skin thoroughly after handling. P280 : Wear protective gloves/ eye protection/ face protection. P302 + P352 : IF ON SKIN: Wash with plenty of water. P337 + P313 : If eye irritation persists: Get medical advice/ attention. P305 + P351 + P338 : IF IN EYES: Rinse cautiously with water for several minutes. Remove contact lenses, if present and easy to do. Continue rinsing. P362 + P364 : Take off contaminated clothing and wash it before reuse. P332 + P313 : If skin irritation occurs: Get medical advice/ attention. |
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Application
AM-251: A Cannabinoid CB1 Receptors (CB1Rs) Antagonist
AM-251 is a cannabinoid CB1 receptors (CB1Rs) antagonist. In areas of the central nervous system (CNS), CB1 receptors have been implicated in regulation of mood and food intake. Reportedly, CB1 agonists increase food intake while CB1 receptor antagonists reduce food intake. AM-251, a CB1 receptor antagonist, have been shown to antidepressant-like and anorectic effects in rats. (The product is for research purpose only.)
References
- Structure-Activity Relationships of Pyrazole Derivatives as Cannabinoid Receptor Antagonists
- Antiobesity effects of chronic cannabinoid CB1 receptor antagonist treatment in diet-induced obese mice
- Antidepressant-like and anorectic effects of the cannabinoid CB1 receptor inverse agonist AM251 in mice
- Inverse agonism and neutral antagonism at cannabinoid CB1 receptors (a review)
- Pharmacological actions of cannabinoids (a review)
PubMed Literature
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